Antagonist Pharmacotherapies for Cannabis Use Disorder

Introduction

  • This article is based on the ASAM Review of Potential Pharmacological Treatments for Cannabis Abuse published on August 9,2021.

  • Antagonist therapies aim to block CB1 receptors. As a result this blocks the action of THC.

  • The equivalent to this strategy is Naltrexone for opioids.

Rimonabant

  • CB1 Antagonist.

  • Early human lab studies showed subjective reduction in “High” after cannabis administration.

  • When studied as a potential treatment for obesity it was discovered that Rimonabant led to increased anxiety, depression and suicidality.

Partial Antagonist

  • Currently under development.

  • Attempt to decrease the subjective effects of cannabis but avoid anxiety, depression, and SI side effects.

References

  1. American Society of Addiction Medicine. (2021, August 9). A review of potential pharmacological treatments for cannabis abuse. https://www.asam.org/blog-details/article/2021/08/09/a-review-of-potential-pharmacological-treatments-for-cannabis-abuse

Agonist Pharmacotherapies for Cannabis Use Disorder

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